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SERD SHR9549

An orally available selective estrogen receptor degrader/downregulator (SERD), with potential antineoplastic activity. Upon oral administration, SERD SHR9549 specifically targets and binds to the estrogen receptor (ER) and induces a conformational change that promotes ER degradation. This prevents ER-mediated signaling and inhibits both the growth and survival of ER-expressing cancer cells.

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Synonym:	selective estrogen receptor degrader SHR9549 selective estrogen receptor downregulator SHR9549
Code name:	SHR 9549 SHR-9549 SHR9549

SERD SHR9549

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